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75438-57-2

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75438-57-2

Moxonidine
Structure Moxonidine
Cat No. SBT1008
Product Name Moxonidine
CAS No. 75438-57-2
Molecular Formula C9H12ClN5O
Molecular Weight 241.68
Purity 99% Min.
Usage 莫索尼啶,又名莫索尼定,化學(xué)名為4-氯-N-(4,5-二氫-1H-咪唑-2-基)-6-甲氧基-2-甲基-5-嘧啶胺,是一高度選擇性咪唑啉-Ⅰ型受體激動(dòng)劑,通過(guò)激動(dòng)Chemicalbook延髓腹外側核(RVLM)-Ⅰ型咪唑啉受體使外周交感神經(jīng)的活性降低,從而舒張血管和減少外周阻力血管阻力使血壓下降,屬于一種新型降壓藥,常用于用于原發(fā)性高血壓的治療。
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