Structure | ![]() |
Cat No. | SBT1003 |
Product Name | Talazoparib(BMN 673) |
Synonym | (8S,9R)-5-Fluoro-8-(4-fluorophenyl)-9-(1-methyl-1H-1,2,4-triazol-5-yl)-8,9-dihydro-2H-pyrido[4,3,2-de]phthalazin-3(7H)-one |
CAS No. | 1207456-01-6 |
Molecular Formula | C19H14F2N6O |
Molecular Weight | 380.35 |
Purity | 99% |
Usage | Talazoparib (BMN 673)是一種新型的PARP抑制劑,IC50為0.58 nM,也有效抑制PARP-2,但不抑制PARG,對PTEN突變型高度敏感。 |
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