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1207456-01-6

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1207456-01-6

Talazoparib(BMN 673)
Structure Talazoparib(BMN 673)
Cat No. SBT1003
Product Name Talazoparib(BMN 673)
Synonym (8S,9R)-5-Fluoro-8-(4-fluorophenyl)-9-(1-methyl-1H-1,2,4-triazol-5-yl)-8,9-dihydro-2H-pyrido[4,3,2-de]phthalazin-3(7H)-one
CAS No. 1207456-01-6
Molecular Formula C19H14F2N6O
Molecular Weight 380.35
Purity 99%
Usage Talazoparib (BMN 673)是一種新型的PARP抑制劑,IC50為0.58 nM,也有效抑制PARP-2,但不抑制PARG,對PTEN突變型高度敏感。
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